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Vastarel

Trimetazidine

Formulated to alleviate coronary myocardial ischaemia to support cardiac oxygen efficiency and target stable angina.

Active ingredient
Trimetazidine
Route
Oral use
Form
Tablet
Strengths
20mg

Prescription and consultation requirements for Vastarel vary by destination and are determined by the fulfilment partner.

Vastarel details

Alternative names
trimetazidine
Therapeutic class
Anti-ischaemic Agent
Pharmacological class
Fatty Acid Oxidation Inhibitor
Known off-label uses
vertigo; tinnitus
Contraindications
parkinson's disease; uncontrolled extrapyramidal symptoms; severe renal failure
Minor side effects
nausea; headache; dizziness
Moderate side effects
indigestion; mild rash; diarrhoea
Serious side effects
drug-induced parkinsonism, requires immediate medical attention
Dosage forms
Tablet
Administration route
Oral use
Supply category
Prescription-only medicine (POM)
Manufacturer
Servier
Onset Time
1–2 weeks
Duration
12–24 hours
Storage instructions
Store below 25°C.
Age restrictions
Approved for adults.
Patient summary

formulated to alleviate coronary myocardial ischaemia to support cardiac oxygen efficiency and target stable angina.

Mechanism of action

Blocks long-chain 3-ketoacyl-CoA thiolase, shifting myocardial metabolism from fatty acid to glucose oxidation to preserve energy.

Pregnancy and breastfeeding

TGA Category C: Use if potential benefits outweigh risks. Breastfeeding: Consult a doctor.